英文名称 | Tariquidar | XR9576 |
---|---|
中文名称 | 他立喹达 |
CAS号 | 206873-63-4 |
分子式 | C38H38N4O6 |
分子量 | 646.73 |
外观 | Off-white to yellow powder |
储存条件 | Store in a dry and dark sealed container, short-term (weeks to months) storage at 0-4 ℃, long-term (months to years) storage at -20 ℃. |
英文名称 | Tariquidar | XR9576 |
---|---|
中文名称 | 他立喹达 |
CAS号 | 206873-63-4 |
分子式 | C38H38N4O6 |
分子量 | 646.73 |
外观 | Off-white to yellow powder |
储存条件 | Store in a dry and dark sealed container, short-term (weeks to months) storage at 0-4 ℃, long-term (months to years) storage at -20 ℃. |
Tariquidar (XR9576) is a potent and specific inhibitor of P-glycoprotein (P-gp) with the high affinity (Kd=5.1 nM).
PMID: 26621623 PMCID: PMC4750702 DOI: 10.1128/AAC.02317-15
PMID: 26661162 PMCID: PMC4976744 DOI: 10.1177/0271678X15606459