英文名称 | Talabostat Mesylate | Val-boroPro mesylate | PT100 mesylate |
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中文名称 | PT100 甲磺酸盐 | [(2R)-1-[(2S)-2-氨基-3-甲基丁酰基]吡咯烷-2-基]硼酸甲磺酸盐 |
CAS号 | 150080-09-4 |
分子式 | C10H23BN2O6S |
分子量 | 310.18 |
外观 | White to off-white powder |
储存条件 | 4°C, sealed storage, away from moisture |
英文名称 | Talabostat Mesylate | Val-boroPro mesylate | PT100 mesylate |
---|---|
中文名称 | PT100 甲磺酸盐 | [(2R)-1-[(2S)-2-氨基-3-甲基丁酰基]吡咯烷-2-基]硼酸甲磺酸盐 |
CAS号 | 150080-09-4 |
分子式 | C10H23BN2O6S |
分子量 | 310.18 |
外观 | White to off-white powder |
储存条件 | 4°C, sealed storage, away from moisture |
Talabostat (Val-boroPro, PT-100) is a dipeptidyl peptidase inhibitor with IC50 values of <4 nM, 4 nM, 11 nM, 310 nM, 560 nM and 390 nM for DPP-IV, DPP8, DPP9, QPP, FAP and PEP respectively. It has antineoplastic and hematopoiesis- stimulating activities.